Immobilization of Benzocaine in Polymeric Nanocontainers. Pharmacokinetic Modeling
- Авторлар: Shkurenko G.Y.1, Lyrshchikov S.Y.1, Gorlov A.A.1, Al’tshuler O.G.1,2, Al’tshuler G.N.1
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Мекемелер:
- Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences
- Kemerovo State University
- Шығарылым: Том 52, № 5 (2018)
- Беттер: 464-466
- Бөлім: Drug Synthesis Methods and Manufacturing Technology
- URL: https://bakhtiniada.ru/0091-150X/article/view/245249
- DOI: https://doi.org/10.1007/s11094-018-1840-3
- ID: 245249
Дәйексөз келтіру
Аннотация
The possibility of immobilizing benzocaine in polymeric nanocontainers made of sulfonated cation exchangers, i.e., sulfonated polycalixarene and KU-23 30/100, was studied. The desorption kinetics of neutral and cationic benzocaine from the polymeric nanocontainers provided the desired drug-release pharmacokinetics upon peroral administration.
Авторлар туралы
G. Shkurenko
Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences
Email: altshulerh@gmail.com
Ресей, 18 Prosp. Sovetskii, Kemerovo, 650000
S. Lyrshchikov
Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences
Email: altshulerh@gmail.com
Ресей, 18 Prosp. Sovetskii, Kemerovo, 650000
A. Gorlov
Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences
Email: altshulerh@gmail.com
Ресей, 18 Prosp. Sovetskii, Kemerovo, 650000
O. Al’tshuler
Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences; Kemerovo State University
Хат алмасуға жауапты Автор.
Email: altshulerh@gmail.com
Ресей, 18 Prosp. Sovetskii, Kemerovo, 650000; 6 Krasnaya St., Kemerovo, 650043
G. Al’tshuler
Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences
Email: altshulerh@gmail.com
Ресей, 18 Prosp. Sovetskii, Kemerovo, 650000
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