Immobilization of Benzocaine in Polymeric Nanocontainers. Pharmacokinetic Modeling


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The possibility of immobilizing benzocaine in polymeric nanocontainers made of sulfonated cation exchangers, i.e., sulfonated polycalixarene and KU-23 30/100, was studied. The desorption kinetics of neutral and cationic benzocaine from the polymeric nanocontainers provided the desired drug-release pharmacokinetics upon peroral administration.

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G. Shkurenko

Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences

Email: altshulerh@gmail.com
俄罗斯联邦, 18 Prosp. Sovetskii, Kemerovo, 650000

S. Lyrshchikov

Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences

Email: altshulerh@gmail.com
俄罗斯联邦, 18 Prosp. Sovetskii, Kemerovo, 650000

A. Gorlov

Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences

Email: altshulerh@gmail.com
俄罗斯联邦, 18 Prosp. Sovetskii, Kemerovo, 650000

O. Al’tshuler

Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences; Kemerovo State University

编辑信件的主要联系方式.
Email: altshulerh@gmail.com
俄罗斯联邦, 18 Prosp. Sovetskii, Kemerovo, 650000; 6 Krasnaya St., Kemerovo, 650043

G. Al’tshuler

Institute of Coal Chemistry and Materials Science, Federal Research Center of Coal and Coal Chemistry, Siberian Branch, Russian Academy of Sciences

Email: altshulerh@gmail.com
俄罗斯联邦, 18 Prosp. Sovetskii, Kemerovo, 650000

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